List of combined sex-hormonal preparations

This is a list of known combined sex-hormonal formulations. Brand names and developmental code names are in parentheses.

• Nandrolone decanoate/nandrolone phenylpropionate (Dinandrol)
• Testosterone propionate/testosterone isocaproate/testosterone caproate (Androteston PP)¹
• Testosterone propionate/testosterone enanthate/testosterone undecylenate (Durasteron)
• Testosterone propionate/testosterone enanthate (Testoviron Depot)
• Testosterone propionate/testosterone ketolaurate (Testosid Depot)
• Testosterone propionate/testosterone phenylpropionate/testosterone isocaproate (Sustanon 100)
• Testosterone propionate/testosterone phenylpropionate/testosterone isocaproate/testosterone caproate (Omnadren 250)
• Testosterone propionate/testosterone phenylpropionate/testosterone isocaproate/testosterone decanoate (Sustanon 250)
• Testosterone propionate/testosterone valerate/testosterone undecylenate (Triolandren)
• Testosterone propionate/testosterone cypionate/prasterone (Sten)

• Boldenone acetate/boldenone cypionate/boldenone propionate/boldenone undecylenate (Equilon 100)
• Testosterone acetate/testosterone undecanoate/testosterone valerate (Deposterona)

• Conjugated estriol (Emmenin, Progynon)
• Conjugated estrogens (Premarin)
• Esterified estrogens (Estratab, Menest)
• Estradiol/estrone/estriol (Hormonin)
• Ethinylestradiol/dienestrol (Foxinette)

• Estradiol benzoate/estradiol phenylpropionate (Dimenformon Prolongatum)

• Estradiol/estradiol enanthate

• Progesterone/hydroxyprogesterone heptanoate/α-tocopherol palmitate (Tocogestan)

• Chlorotrianisene/methyltestosterone (Tace mit Androgen)¹
• Conjugated estrogens/methyltestosterone (Premarin with Methyltestosterone)
• Dienestrol/methyltestosterone (Estan, Lucidon)
• Dienestrol diacetate/methyltestosterone (Farmatest)
• Diethylstilbestrol/methyltestosterone (Tylosterone)
• Esterified estrogens/methyltestosterone (Covaryx, Eemt, Essian, Estratest, Menogen, Syntest)
• Ethinylestradiol/methyltestosterone (Climatone, Dumone, Duotrone, Estandron, Femandren, Femovirin, Gynetone, Lynandron, Mepilin, Mixogen, Primodian)¹²
• Methylestradiol/methyltestosterone (Klimanosid)²
• Methylestradiol/methyltestosterone/reserpine (Klimanosid R)¹

• Estradiol benzoate/testosterone propionate (Bothermon)
• Estradiol benzoate/estradiol dienanthate/testosterone enanthate benzilic acid hydrazone (Climacteron, Lactimex, Lactostat)
• Estradiol benzoate/estradiol phenylpropionate/testosterone propionate/testosterone phenylpropionate/testosterone isocaproate (Estandron Prolongatum, Lynandron Prolongatum, Mixogen [Injection])
• Estradiol benzoate/testosterone isobutyrate (Femandren M, Folivirin)
• Estradiol butyrylacetate/testosterone ketolaurate/reserpine (Klimanosid R-Depot)
• Estradiol cypionate/testosterone cypionate (Depo-Testadiol, Femovirin)
• Estradiol cypionate/testosterone enanthate (Supligol)
• Estradiol valerate/prasterone enanthate (Binodian Depot, Cidodian Depot, Gynodian Depot, Klimax, Supligol NF)
• Estradiol valerate/testosterone enanthate (Deladumone, Despamen, Ditate, Ditate-DS, Gravignost, Primodian Depot, Valertest)

• Diethylstilbestrol/methyltestosterone (Maxymin, Tylosterone)
• Diethylstilbestrol/testosterone (Rapigain)
• Estradiol benzoate/estradiol enanthate/testosterone enanthate (Uni-Bol)
• Estradiol benzoate/testosterone propionate (Component E-H, Implix BF, Progro H, Synovex H)
• Ethinylestradiol/methyltestosterone (Taril)

In birth control pills:

• Drospirenone/estetrol (Nextstellis, Drovelis, Lydisilka)
• Estradiol/nomegestrol acetate (Naemis, Zoely)
• Estradiol valerate/cyproterone acetate (Femilar)
• Estradiol valerate/dienogest (Natazia, Qlaira)
• Ethinylestradiol/chlormadinone acetate (Belara)³
• Ethinylestradiol/cyproterone acetate (Diane, Diane-35)
• Ethinylestradiol/desogestrel (Alenvona, Apri,⁴ Azurette,⁵ Bekyree,⁶ Bimizza,⁷ Caziant,⁸ Cesia,⁹ Cimizt,¹⁰ Cyclessa,¹¹ Cyred,¹² Denise, Desogen,¹³ Desirett, Emoquette,¹⁴ Enskyce,¹⁵ Gedarel, Gracial, Isibloom,¹⁶ Juleber,¹⁷ Kalliga, Kariva,¹⁸ Kimidess,¹⁹ Laurina, Linessa, Marvelon,²⁰²¹²² Mercilon,²³²⁴ Mircette,²⁵ Mirvala, Novynette, Ortho-Cept,²⁶ Pimtrea,²⁷ Reclipsen,²⁸ Regulon, Simliya,²⁹ Solia, Velivet,³⁰ Viorele,³¹ Volnea³²)
• Ethinylestradiol/dienogest (Valette)
• Ethinylestradiol/dimethisterone (Oracon)
• Ethinylestradiol/drospirenone (Yasmin, Yasminelle, Yaz)
• Ethinylestradiol/drospirenone/levomefolic acid (Beyaz, Safyral)
• Ethinylestradiol/etynodiol diacetate (Demulen)
• Ethinylestradiol/gestodene (Femodene, Femodette, Gynera, Harmonet, Meliane, Minesse, Minulet)
• Ethinylestradiol/levonorgestrel (Amethyst, Aviane, Balcoltra, Falmina, Levlen, Lillow, Orsythia, Vienva)
• Ethinylestradiol/levonorgestrel/bisglycinate
• Ethinylestradiol/levonorgestrel/ferrous fumarate
• Ethinylestradiol/lynestrenol (Lyndiol)
• Ethinylestradiol/medroxyprogesterone acetate (Gianda, Provest)
• Ethinylestradiol/megestrol acetate (Nuvacon, Volidan)
• Ethinylestradiol/norethisterone (Brevicon, Norinyl 1+35, Ortho-Novum 7/7/7, Taytulla, Tri-Norinyl, Zenchent)
• Ethinylestradiol/norethisterone/ferrous fumarate (Blisovi 24 FE, Estrostep Fe, Femcon FE, Kaitlib FE, Lo Minastrin Fe, Loestrin 24 Fe, Microgestin 24 FE)
• Ethinylestradiol/norethisterone acetate (FemHRT)
• Ethinylestradiol/norethisterone acetate/ferrous fumarate
• Ethinylestradiol/norgestimate (Ortho Tri-Cyclen, Sprintec)
• Ethinylestradiol/norgestrel (Ovral)
• Ethinylestradiol/norgestrienone (Miniplanor, Planor)
• Ethinylestradiol/quingestanol acetate (Riglovis)
• Ethinylestradiol sulfonate/norethisterone acetate (Deposiston)
• Mestranol/anagestone acetate (Neo-Novum)
• Mestranol/chlormadinone acetate (C-Quens, Lutedion)
• Mestranol/etynodiol diacetate (Ovulen)
• Mestranol/hydroxyprogesterone acetate (Hormolidin)
• Mestranol/lynestrenol (Lyndiol)
• Mestranol/norethisterone (Norethin, Noriday, Norinyl, Norquen, Ortho-Novum)
• Mestranol/noretynodrel (Enavid, Enovid)
• Quinestrol/etynodiol diacetate (Soluna)
• Quinestrol/levonorgestrel (Yuèkětíng, Àiyuè)
• Quinestrol/norgestrel (Compound Norgestrel)
• Quinestrol/quingestanol acetate (Unovis)

For menopausal hormone therapy and/or gynecological disorders:

• Conjugated estrogens/medrogestone (Presomen)
• Conjugated estrogens/medroxyprogesterone acetate (Prempro, Premphase)
• Conjugated estrogens/norgestrel (Prempak-C)
• Estradiol/drospirenone (Angeliq)
• Estradiol/dydrogesterone (Femoston)
• Estradiol/gestodene (Avaden, Avadene)
• Estradiol/levonorgestrel
• Estradiol/medroxyprogesterone acetate (Indivina, Tridestra)
• Estradiol/norethisterone acetate (Activella, Activelle, Cliane, Estalis, Eviana, Evorel, Kliogest, Novofem)
• Estradiol/norgestimate (Prefest)
• Estradiol/progesterone (Bijuva)
• Estradiol/trimegestone (Lovelle, Totelle)
• Estradiol valerate/cyproterone acetate (Climen, Climen 28)
• Estradiol valerate/estriol/levonorgestrel (CycloÖstrogynal)
• Estradiol valerate/levonorgestrel (Cyclo-Progynova N)
• Estradiol valerate/medroxyprogesterone acetate (Dilena, Divina, Divitren, Farludiol, Indivina, Sisare)
• Estradiol valerate/norethisterone (Climagest, Climesse)
• Estradiol valerate/norethisterone acetate (Cliovelle, Norestin, Trisequens)
• Estradiol valerate/norgestrel (Cyclacur, Cyclocur, Cyclo-Progynova, Postoval, Progyluton)
• Ethinylestradiol/ethisterone (Amenorone, Di-Pro, Duosterone, Menstrogen, Oracecron, Orasecron)²¹
• Mestranol/noretynodrel (Enovid)

In birth control pills:

• Estradiol/norethisterone (Netagen, Netagen 403)

In contraceptive patches:

• Ethinylestradiol/norelgestromin (Evra, Ortho Evra, Xulane)

For menopausal hormone therapy:

• Estradiol/levonorgestrel (Climara Pro)
• Estradiol/norethisterone acetate (CombiPatch)

In contraceptive vaginal rings:

• Ethinylestradiol/etonogestrel (Circlet, NuvaRing)
• Segesterone acetate/ethinylestradiol (Annovera)

In combined injectable contraceptives:

• Estradiol/megestrol acetate (Mego-E, Chinese Injectable No. 2)
• Estradiol benzoate/estradiol valerate/hydroxyprogesterone caproate (Sin-Ol)
• Estradiol benzoate butyrate/algestone acetophenide (Redimen, Soluna, Unijab)
• Estradiol cypionate/hydroxyprogesterone caproate (Sinbios)
• Estradiol cypionate/medroxyprogesterone acetate (Cyclo-Provera, Cyclofem, Lunelle)
• Estradiol enanthate/algestone acetophenide (Anafertin, Deladroxate, Perlutan, Topasel, Yectames)
• Estradiol valerate/hydroxyprogesterone caproate (Chinese Injectable No. 1)
• Estradiol valerate/norethisterone enanthate (Mesigyna, Mesygest)

For menopausal hormone therapy, gynecological disorders, habitual abortion, and other indications:

• Estradiol/progesterone (Juvenum)
• Estradiol benzoate/hydroxyprogesterone caproate (Primosiston)
• Estradiol benzoate/progesterone (Duogynon, Sistocyclin)
• Estradiol dipropionate/hydroxyprogesterone caproate (EP Hormone Depot)
• Estradiol hemisuccinate/progesterone (Hosterona)
• Estradiol pivalate/progesterone (Estrotate with Progesterone)
• Estradiol valerate/hydroxyprogesterone caproate (Gravibinan, Gravibinon)
• Estrone/progesterone (Synergon)

In combined injectable contraceptives:

• Estradiol/progesterone (in microspheres and macrocrystalline aqueous suspension)
• Estradiol undecylate/norethisterone enanthate
• Estradiol valerate/megestrol acetate
• Estradiol valerate/methenmadinone caproate (Lutofollin)
• Polyestradiol phosphate/medroxyprogesterone acetate
• Additional preparations listed at Combined injectable birth control § Research

For other indications:

• Estradiol valerate/gestonorone caproate (SH-834, SH-8.0834)

• Estradiol benzoate/progesterone (Component E-S, Implix BM, Synovex C, Synovex S)
• Estradiol valerate/norgestomet (Syncro-Mate-B)

• Methyltestosterone/ethisterone (Androgeston)¹

• Testosterone propionate/progesterone (Testoluton)^33123435

• Danazol/megestrol acetate (Dogalact)
• Nandrolone decanoate/methandriol dipropionate (Filybol, Tribolin)
• Nandrolone phenylpropionate/methandriol dipropionate (RWR)

• Methylestradiol/normethandrone (Ginecosid, Ginecoside, Mediol, Renodiol)

• Ethinylestradiol/drospirenone/prasterone

• Estradiol/progesterone/methyltestosterone (Trihormonal)¹
• Ethinylestradiol/ethisterone/methyltestosterone (Trinestryl, Trimone Sublets)¹

• Estradiol benzoate/progesterone/methandriol dipropionate (Progestandron)
• Estradiol benzoate/progesterone/testosterone propionate (Lukestra, Steratrin, Trihormonal, Trinestryl)¹²³⁶
• Estradiol benzoate/estradiol valerate/norethisterone acetate/testosterone enanthate (Ablacton)
• Estradiol dibutyrate/hydroxyprogesterone heptanoate/testosterone caproate (Triormon Depositum)
• Estradiol diundecylate/hydroxyprogesterone heptanoate/testosterone cyclohexylpropionate (Trioestrine Retard)
• Estradiol hexahydrobenzoate/hydroxyprogesterone caproate/testosterone hexahydrobenzoate (Trinestril AP)
• Estrone/progesterone/testosterone (Tristeron, Tristerone)³⁶

• Estrapronicate/hydroxyprogesterone heptanoate/nandrolone undecanoate (Trophobolene, Trophoboline)

• Estradiol/trenbolone acetate (Component, Compudose-G, Progro TE-H, Revalor, Synovex)
• Estradiol benzoate/trenbolone acetate (Synovex Choice, Synovex One, Synovex Plus, Synovex with Trenbolone Acetate)

• Conjugated estrogens/bazedoxifene (Duavee)

• Esterified estrogens/raloxifene
• Estradiol/raloxifene

• Estradiol benzoate/prednisolone/salicylic acid (Alpicort E, Alpicort F, Alpicort Plus)

• Estradiol benzoate/gentamicin/hydrocortisone/nystatin (Cridermol Fem, Ginabiot, Ginecovan)
• Estradiol benzoate/monalazone (Malun-25)

• Goserelin/bicalutamide (ZolaCos CP)
• Leuprorelin/norethisterone acetate (Lupaneta Pack)

See also

See also

• List of sex-hormonal medications available in the United States
• List of sex-hormonal aqueous suspensions
• List of steroid esters
• List of marketed estradiol benzoate formulations

References

References

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